|


The Royal Society of Chemistry 1st May 2007 - High Throughput Medicinal Chemistry
    
High throughput techniques have revolutionised the drug discovery process and are widely used in medicinal
chemistry to speed the development of new and higher quality drug candidates. The scientific programme of
the "High Throughput Medicinal Chemistry" meeting will include presentations on computational tools,
purification of small organic molecules, ADME , fragment based design and case studies from GlaxoSmithKline,
AstraZeneca and Merck Sharpe and Dohme.
Date: |
1st May 2007 |
Location: |
SC1 auditorium, GlaxoSmithKline, Harlow |
Application and Fees: |
RSC Members - £112.00, Non RSC Members - £153.00 |
For Further Information: |
Please contact Michele Sahrle. |
|
 |
 |
09:00 |
Registration and Coffee |
09:50 |
Introduction |
10:00 |
Microwaves and Microreactors: New Faster Methods in Heterocyclic Chemistry Mark Bagley, Cardiff University |
10:40 |
The Application of High Throughput Chemistry in Discovery Research: Hope, Hype and Reality Chris Hill, Organon |
11:20 |
Asymmetric Catalysis: Simple and Easy! Prof. Carsten Bolm, RWTH, Aachen University, Aachen, Germany |
12:00 |
Tour of High Throughput Chemistry Facility and lunch |
13:15 |
The Use of Combinatorial and Parallel Synthesis for Lead Identification and Optimisation Brian McKittrick, Schering-Plough, NJ |
13:55 |
Fragment based approaches to drug discovery John Reader, Sareum Ltd |
14:35 |
Design of Novel Matrix Metalloprotease Inhibitors - Classical Structure Based Design Using High Throughput Techniques Ian Holmes, GSK |
15:15 |
Tea and Coffee |
15:40 |
Metalated Flatland Motifs for Pharmaceutical Research and Development Prof. Victor Snieckus, Queen's University, Kingston, Canada |
16:20 |
The Changing Face of Chemistry in Drug Discovery David A Roberts, AstraZeneca |
17:00 |
Close Meeting / Wine Reception |
19:00 |
finish |
|
|
 |
 |
|